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| CAS No. | 72956-09-3 |
| Chemical Name: | Carvedilol |
| Synonyms: | COREG;Carca;Kredex;Querto;Artist;Carloc;Carvas;DQ-2466;Artione;Cadilan |
| CBNumber: | CB8351959 |
| Molecular Formula: | C24H26N2O4 |
| Formula Weight: | 406.47 |
| MOL File: | 72956-09-3.mol |
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| Carvedilol Property |
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| storage temp. : |
Store at +4°C |
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Carvedilol Chemical Properties,Usage,Production |
Chemical Properties
Colourless Crystalline Solid |
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Usage
A nonselective -adrenergic blocker with a1-blocking activity. An antihypertensive used in the treatment of congestive heart failure.
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Usage
Carvedilol is a nonselective β-adrenergic blocker with α1-blocking activity. Carvedilol is an antihypertensive used in the treatment of congestive heart failure. |
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Usage
For the treatment of mild or moderate (NYHA class II or III) heart failure of ischemic or cardiomyopathic origin. |
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Biological Activity
Potent β -adrenoceptor and α 1 -adrenoceptor antagonist (K i values are 0.81, 0.96 and 2.2 nM for β 1 -, β 2 - and α 1 -adrenoceptors respectively) that displays antihypertensive and peripheral vasodilatory activity. Blocks cardiac inward-rectifier K + (K IR ) channels, voltage-dependent Ca 2+ channels and exhibits antioxidant properties at higher concentrations. |
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| Carvedilol Preparation Products And Raw materials |
Raw materials
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Preparation Products
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| Carvedilol Suppliers Global( 162)Suppliers |
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