PROXYFAN MALEATE Property |
storage temp. : |
Desiccate at RT |
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PROXYFAN MALEATE Chemical Properties,Usage,Production |
Biological Activity
High affinity histamine H 3 receptor ligand (pK i = 8.62) that acts as a protean agonist at recombinant and native receptors. In functional studies, activity ranges from full agonist to inverse agonist depending on system used. Displays partial agonist effects on cAMP inhibition and MAPK activity, neutral antagonist activity on histamine release and partial inverse agonism of [ 3 H]-arachidonic acid release. |
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PROXYFAN MALEATE Preparation Products And Raw materials |
Raw materials
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Preparation Products
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PROXYFAN MALEATE Suppliers Global( 4)Suppliers |
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