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CAS No. | 106243-16-7 |
Chemical Name: | THIOPERAMIDE MALEATE |
Synonyms: | Thiop;MR 12842;thioperamide;THIOPERAMIDE MALEATE;THIOPERAMIDE MALEATE SALT;THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE;N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide;N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide;N-CYCLOHEXYL-4-(IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE;N-CYCLOHEXYL-4-(1H-IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE |
CBNumber: | CB5245732 |
Molecular Formula: | C19H28N4O4S |
Formula Weight: | 408.52 |
MOL File: | 106243-16-7.mol |
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THIOPERAMIDE MALEATE Property |
storage temp. : |
Store at -20°C |
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solubility : |
H2O: 10 mg/mL
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THIOPERAMIDE MALEATE Chemical Properties,Usage,Production |
Biological Activity
Potent histamine H 3 and H 4 antagonist/inverse agonist. K i values are 25 and 27 nM for human recombinant H 3 and H 4 receptors respectively. Blocks eosinophil shape change (IC 50 = 1.4 μ M) and chemotaxis (IC 50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H 3 Receptor Tocriset™ . |
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THIOPERAMIDE MALEATE Preparation Products And Raw materials |
Raw materials
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Preparation Products
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THIOPERAMIDE MALEATE Suppliers Global( 19)Suppliers |
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106243-16-7(THIOPERAMIDE MALEATE)Related Search: |
1,3-Dibutyl-2-thiourea
1-CYCLOHEXYL-2-THIOUREA
4-(1H-IMIDAZOL-4-YL)-1-METHYL-PIPERIDINE
4-(1H-IMIDAZOLE-4(5)-YL) PIPERIDINE
N,N-DIETHYLTHIOUREA
1-PIPERIDINETHIOCARBOXAMIDE
THIOPERAMIDE MALEATE
N,N'-DI-N-PROPYLTHIOUREA
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thioperamide
106243-16-7
N-CYCLOHEXYL-4-(IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
N-CYCLOHEXYL-4-(1H-IMIDAZOL-4-YL)-1-PIPERIDINECARBOTHIOAMIDE MALEATE
MR 12842
THIOPERAMIDE MALEATE
THIOPERAMIDE MALEATE SALT
Potent and selective H3 histamine receptor antagonist that crosses the blood-brain barrier.
THIOPERAMIDE MALEATE (MR 12842) POTENT A ND SELECTIVE
C15H24N4SC4H4O4
Histamine receptor
N-Cyclohexyl-4-(1H-imidazol-4-yl)-1-piperidinecarbothioamide
Thiop
Histamine
N-Cyclohexyl-4-(imidazol-4-yl)-1-piperidinecarbothioamide
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