3-MATIDA Property |
storage temp. : |
Store at +4°C |
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3-MATIDA Chemical Properties,Usage,Production |
Biological Activity
Potent metabotropic glutamate mGlu 1 receptor antagonist (IC 50 = 6.3 μ M at rat mGlu 1a ). Displays ≥ 40-fold selectivity over other receptors: mGlu 5 , mGlu 2 , mGlu 4a (IC 50 > 300 μ M), NMDA and AMPA (IC 50 = 250 μ M). Neuroprotective in cultured murine cortical cells and rat hippocampal slice cultures in vitro . Reduces the volume of ischemia-induced brain infarcts in rats following systemic administration in vivo . |
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3-MATIDA Preparation Products And Raw materials |
Raw materials
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Preparation Products
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3-MATIDA Suppliers Global( 5)Suppliers |
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