AMINOPURVALANOL A Property |
storage temp. : |
Store at +4°C |
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AMINOPURVALANOL A Chemical Properties,Usage,Production |
Biological Activity
Cell-permeable cyclin-dependent kinase inhibitor. IC 50 values are 0.033, 0.033, 0.028 and 0.020 μ M for cdk1/cyclin B, cdk2/cyclin A, cdk2/cyclin E, and cdk5/p35 respectively. Inhibits ERK1 (IC 50 = 12.0 μ M) and ERK2 (IC 50 = 3.1 μ M) and is 3000-fold selective over a range of other protein kinases (IC 50 > 100 μ M). Arrests cell cycle at G 2 /M boundary (IC 50 = 1.25 μ M), and induces apoptosis at concentrations > 10 μ M. |
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AMINOPURVALANOL A Preparation Products And Raw materials |
Raw materials
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Preparation Products
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AMINOPURVALANOL A Suppliers Global( 8)Suppliers |
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