AM 251

CAS No.	183232-66-8
Chemical Name:	AM 251
Synonyms:	AM 251;AM-251 ,99%;AM 251 (pharmaceutical);1-(2,4-DICHLOROPHENYL)-5-(4-IODOPHENYL)-4-METHYL-N-1-PIPERIDINYL-1 H-PYRAZOLE-3-CARBOXAMIDE;1H-Pyrazole-3-carboxamide, 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-;N-(PIPERIDIN-1-YL)-5-(4-IODOPHENYL)-1-(2,4-DICHLOROPHENYL)-4-METHYL-1H-PYRAZOLE-3-CARBOXAMIDE;1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide AM251
CBNumber:	CB2169367
Molecular Formula:	C22H21Cl2IN4O
Formula Weight:	555.24
MOL File:	183232-66-8.mol

AM 251 Property

mp :

195-196℃

storage temp. :

Store at RT

solubility :

DMSO: >10 mg/mL, soluble

form :

solid

color :

white

Safety

Hazard Codes :

Risk Statements :

36/37/38

Safety Statements :

26-36

WGK Germany :

AM 251 Chemical Properties,Usage,Production

Chemical Properties
White to Off-White Solid

Usage
Inhibitor of CB1 receptors. AM 251is a biarylpyrazole compound which has been considered for many years as the prototypical cannabinoid (CB) receptor antagonist

Biological Activity
Potent CB 1 receptor antagonist (IC 50 = 8 nM, K i = 7.49 nM) that displays 306-fold selectivity over CB 2 receptors. Also potent GPR55 agonist (EC 50 = 39 nM). Also available as part of the Cannabinoid CB 1 Receptor Tocriset™ .

AM 251 Preparation Products And Raw materials

Raw materials

Preparation Products

AM 251 Suppliers Global( 37)Suppliers

Supplier	Tel	Fax	Email	Country	ProdList	Advantage
J & K SCIENTIFIC LTD.	--	--	jkinfo@jkchemical.com;market3@jkchemical.com	CHINA	96847	76
3B Pharmachem (Wuhan) International Co.,Ltd.	86-21-50328103 * 801、802、803、804 Mobile:18930552037	86-21-50328109	67055399@qq.com	CHINA	15983	69
Ascent Scientific	4401179829988	4402030 700 369	customerservice@ascentscientific.co.uk	UNITED KINGDOM	282	60
VDM Biochemicals	0330-2528181	0330-2528171	sales@vdmbio.com	USA	511	64
Chemsky（shanghai）International Co.,Ltd.	021-50135380		shchemsky@sina.com	CHINA	32553	50
T&W GROUP	+86-21-61551611, 61551413, 61551420, 61551610	+86-21-50676805	contact@trustwe.com	CHINA	13395	58
Shanghai Haoyuan Chemexpress Co., Ltd	86-21-58998590	86-21-53700326, 86-21-58998590	sales@chemexpress.cn	CHINA	10011	61
Shanghai Aladdin Bio-Chem Technology Co.,LTD	021-20337333/400-620-6333	021-50323701	sale@aladdin-e.com	CHINA	24330	65
MedChemexpress LLC	609-228-6898	609-228-5909	sales@medchemexpress.cn	USA	4935	58
AdooQ BioScience, LLC	+1 (866) 930-6790	+1 (866) 333-9607	info@adooq.com	USA	2786	58

183232-66-8(AM 251)Related Search:

Olaparib Pyrazole-3-carboxamide AM 251 TRIFLUOROACETATE AM 251 TRIFLUOROACETATE SALT N-Aminopiperidine hydrochloride AM 251

AM 251 1-(2,4-DICHLOROPHENYL)-5-(4-IODOPHENYL)-4-METHYL-N-1-PIPERIDINYL-1 H-PYRAZOLE-3-CARBOXAMIDE 183232-66-8 N-(PIPERIDIN-1-YL)-5-(4-IODOPHENYL)-1-(2,4-DICHLOROPHENYL)-4-METHYL-1H-PYRAZOLE-3-CARBOXAMIDE C22H21Cl2IN4O C22H21N4OCl2I Cannabinoid receptor Cannabinoid AM-251 ,99% Aromatics Heterocycles Cannabinoids AM 251 (pharmaceutical) 1H-Pyrazole-3-carboxamide, 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl- 1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide AM251