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CAS番号. | 162256-50-0 |
化学名: | |
别名: | |
英語化学名: | CI 1020 |
英語别名: | CI 1020;PD 156707;3-(1,3-Benzodioxol-5-yl)-5-hydroxy-5-(4-methoxyphenyl)-4-[(3,4,5-trimethoxyphenyl)methyl]-2(5H)-furanone |
CBNumber: | CB81873005 |
分子式: | C28H26O9 |
分子量: | 0 |
MOL File: | 162256-50-0.mol |
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CI 1020 化学特性,用途語,生産方法 |
使用
A novel endothelin-A receptor antagonist, in hypoxic pulmonary hypertension. |
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生物活性
Highly selective, orally active, non-peptide endothelin-A receptor (ET A ) antagonist (IC 50 values are 0.3 and 480 nM for ET A and ET B receptors respectively). Antihypertensive; blocks ET-1-induced pressor responses following oral administration. |
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CI 1020 上流と下流の製品情報 |
原材料
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準備製品
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CI 1020 生産企業 Global( 6)Suppliers |
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