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CAS番号. | 183320-51-6 |
化学名: | |
别名: | |
英語化学名: | OSI-420 |
英語别名: | CP-473420;DesMethyl Erlotinib;OSI-420 hydrochloride;OSI-420 (DesMethyl Erlotinib);DesMethyl Erlotinib (CP-473420) HCl;OSI-420 (DesMethyl Erlotinib,CP-473420);Erlotinib O-DesMethyl Metabolite IsoMer (M14) HCl;2-(4-(3-ethynylphenylamino)-7-(2-methoxyethoxy)quinazolin-6-yloxy)ethanol hydrochloride;2-[[4-[(3-Ethynylphenyl)amino]-7-(2-methoxyethoxy)-6-quinazolinyl]oxy]ethanol hydrochloride;Ethanol, 2-[[4-[(3-ethynylphenyl)aMino]-7-(2-Methoxyethoxy)-6-quinazolinyl]oxy]-, hydrochloride |
CBNumber: | CB22561488 |
分子式: | C21H21N3O4.HCl |
分子量: | 0 |
MOL File: | Mol file |
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OSI-420 化学特性,用途語,生産方法 |
使用
OSI-420 (Desmethyl Erlotinib,CP-473420) is an active metabolite of erlotinib which is an orally active EGFR tyrosin kinase inhibitor with IC50 of 2 and 20 nM for the inhibition of human EGFR and EGFR autophosphorylation in tumor cells.
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OSI-420 上流と下流の製品情報 |
原材料
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準備製品
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OSI-420 生産企業 Global( 21)Suppliers |
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