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CAS番号. | 1390637-82-7 |
化学名: | |
别名: | |
英語化学名: | PF-04981517 |
英語别名: | CYP3cide;PF-4981517;PF-04981517;1-Methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-piperidin-1-ylpyrrolidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidine;1H-Pyrazolo[3,4-d]pyrimidine, 1-methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-(1-piperidinyl)-1-pyrrolidinyl]- |
CBNumber: | CB12620906 |
分子式: | C26H32N8 |
分子量: | 456.58588 |
MOL File: | 1390637-82-7.mol |
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PF-04981517 化学特性,用途語,生産方法 |
化学的特性
White to Off-White Solid |
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使用
CYP3cide is a potent and selective time dependent inactivator of Cytochrome P450 3A4 (CYP3A4). CYP3A4 is an important enzymes involved in the metabolism of xenobiotics in the human body and constitutes to about a quarter of all CYPs in the human body. CYP3cide provides a useful in vitro tool in defining the individual roles of CYP3A4 versus CYP3A5 in the metabolism of drugs. |
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PF-04981517 上流と下流の製品情報 |
原材料
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準備製品
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PF-04981517 生産企業 Global( 10)Suppliers |
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