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CAS番号. | 928037-13-2 |
化学名: | |
别名: | |
英語化学名: | Golvatinib (E7050) |
英語别名: | E-7050;Golvatinib;Golvatinib (E7050);E-7050 (Golvatinib);N-[2-Fluoro-4-[[2-[[[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl]amino]pyridin-4-yl]oxy]phenyl]-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide;1,1-Cyclopropanedicarboxamide, N-[2-fluoro-4-[[2-[[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]amino]-4-pyridinyl]oxy]phenyl]-N'-(4-fluorophenyl)-;N-[2-Fluoro-4-[[2-[[[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl]amino]pyridin-4-yl]oxy]phenyl]-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide Golvatinib(E-7050) |
CBNumber: | CB12589746 |
分子式: | C33H37F2N7O4 |
分子量: | 633.6881864 |
MOL File: | 928037-13-2.mol |
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Golvatinib (E7050) 化学特性,用途語,生産方法 |
使用
E7050 is a dual c-Met and VEGFR-2 inhibitor with IC50 of 14 nM and 16 nM, respectively. |
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使用
Golvatinib is a potent and orally available inhibitor of c-MET and VEGFR-2 that exhibits potential antitumor properties by suppressing the overexpression of these receptor tyrosine kinases. |
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Golvatinib (E7050) 上流と下流の製品情報 |
原材料
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準備製品
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Golvatinib (E7050) 生産企業 Global( 28)Suppliers |
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