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CAS No. | 755037-03-7 |
Chemical Name: | Regorafenib |
Synonyms: | Regafenib;regorafinib;BAY 73-4506;Regorafenib;Reggae sorafenib;Fluoro-Sorafenib;Regorafenib C3X-1410;Stivarga(regorafenib);BAY 73-4506(Regorafenib);Regorafenib (BAY 73-4506) |
CBNumber: | CB32498792 |
Molecular Formula: | C21H15ClF4N4O3 |
Formula Weight: | 482.8154128 |
MOL File: | 755037-03-7.mol |
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Regorafenib Chemical Properties,Usage,Production |
Usage
It inhibits PDGFR tyrosine kinase with IC50=83nM. It is useful for the treatment of inflammation and as an anti-proliferative agent. |
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Usage
BAY 73-4506 (Regorafenib) is a multikinase inhibitor with IC50 of 17, 40 and 69 nM c-KIT, VEGFR2, B-Raf. |
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Usage
Regorafenib (BAY 73-4506) is a multi-target inhibitor for VEGFR1, VEGFR2, VEGFR3, PDGFRβ, Kit, RET and Raf-1 with IC50 of 13 nM/4.2 nM/46 nM, 22 nM, 7 nM, 1.5 nM and 2.5 nM, respectively |
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Regorafenib Preparation Products And Raw materials |
Raw materials
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Preparation Products
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Regorafenib Suppliers Global( 118)Suppliers |
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